反应条件
1: With potassium tert-butylate in N,N-dimethyl-formamide T=-5°C; 1 h; Inert atmosphere; 2: in N,N-dimethyl-formamide T=-5°C; 1 h; Inert atmosphere;
参考文献
Doiron, Jeremie; Soultan, Al Haliffa; Richard, Ryan; Toure, Mamadou Mansour; Picot, Nadia; Richard, Remi; Cuperlovic-Culf, Miroslava; Robichaud, Gilles A.; Touaibia, Mohamed
European Journal of Medicinal Chemistry, 2011 , vol. 46, # 9 p. 4010 - 4024