1: 1.39 g / Et2NH, CuI / Pd(OAc)2(PPh3)2 / 20 h / Ambient temperature 2: piperidine, formic acid / Pd(OAc)2(PPh3)2 / dimethylformamide / 20 h / 60 °C View Scheme
参考文献
Arcadi, A.; Cacchi, S.; Marinelli, F.
Tetrahedron, 1985 , vol. 41, # 22 p. 5121 - 5132
1: 1.39 g / Et2NH, CuI / Pd(OAc)2(PPh3)2 / 20 h / Ambient temperature 2: piperidine, formic acid / Pd(OAc)2(PPh3)2 / dimethylformamide / 20 h / 60 °C View Scheme
参考文献
Arcadi, A.; Cacchi, S.; Marinelli, F.
Tetrahedron, 1985 , vol. 41, # 22 p. 5121 - 5132