6-(1-((叔丁基二甲基甲硅烷基)氧基)-2-硝基丙基)-[1,2,4]噻唑并[1,5-a]吡啶合成路线 (共 2 条)
反应条件
1H-imidazole in N,N-dimethyl-formamide T=5 - 20°C;
参考文献
BIOGEN IDEC MA INC.
Patent: WO2008/94556 A2, 2008 ;
Location in patent: Page/Page column 32 ;
反应条件
ammonium formate; palladium on activated carbon in methanol T=5 - 20°C;
参考文献
BIOGEN IDEC MA INC.
Patent: WO2008/94556 A2, 2008 ;
Location in patent: Page/Page column 32 ;