反应条件
1: POCl3 / 2 h / 40 °C
2: 2.) Na2CO3 / 1.) chloroform, reflux, 15 h, 2.) water, 15 min
3: 13 percent / hydrazine hydrate, Raney Nickel / ethanol / 1.) room temperature, 30 min, 2.) reflux, 60 min
View Scheme
参考文献
Mulay, Balbhim D.; Kelkar, Shriniwas L.; Wadia, Murzban S.
Synthetic Communications, 1987 , vol. 17, # 5 p. 535 - 542