1: With lithium aluminium tetrahydride in tetrahydrofuran
3 h; Heating / reflux;
2: With sodium hydroxide; water in tetrahydrofuran
T=0°C;
参考文献
Wong, Norman C.W.; Tucker, Joseph E.L.; Hansen, Henrik C.; Chiacchia, Fabrizio S.; McCaffrey, David
Patent: US2008/188467 A1, 2008 ;
Location in patent: Page/Page column 44 ;
US 20080188467 A1