反应条件
1: trimethylsilyl iodide / 0.5 h / Ambient temperature 2: 2.) CH3OH / 1.) acetonitrile, RT, 3 h, 2.) acetone View Scheme
参考文献
Brown; Kinnick; Morin Jr.; Vasileff; Counter; Davidson; Ensminger; Eudaly; Kasher; Katner; Koehler; Kurz; Lindstrom; Lunn; Preston; Ott; Quay; Shadle; Steinberg; et al.
Journal of Medicinal Chemistry, 1990 , vol. 33, # 8 p. 2114 - 2121