4-(4-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)-3-环己烯)吗啉合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in N,N-dimethyl-formamide T=85°C; 17 h;
参考文献
EISAI R andamp; D MANAGEMENT CO. LTD; GRACZYK, Piotr; BHATIA, Gurpreet, Singh
Patent: WO2010/15803 A1, 2010 ;
Location in patent: Page/Page column 32; 35-36 ;
WO 2010/015803 A1