反应条件
1: 86 percent / CF3COOH, Et3SiH / Ambient temperature 2: 57 percent / K2CO3, NaI / acetone / 15 h / Heating 3: 92 percent / tetrahydrofuran; ethanol; methanol / 12 h / Heating 4: 65 percent / EtSH, BF3*Et2O / 1 h / Ambient temperature View Scheme
参考文献
Chang; Ares; Anderson; Sabol; Wallace; Farooqui; Uretsky; Miller
Journal of Medicinal Chemistry, 1987 , vol. 30, # 1 p. 214 - 218