反应条件
1: NaOAc / pyridine; dimethylformamide / 20 h / Ambient temperature 2: 1.) 15 percent BuLi / 1.) THF/hexane, -70 deg C, 10 min, 2.) -70 deg C, 1 h View Scheme
参考文献
Hofmeister; Annen; Laurent; Petzoldt; Wiechert
Arzneimittel-Forschung/Drug Research, 1986 , vol. 36, # 5 p. 781 - 783