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Wenner; Plati
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Gault; Viout
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1: 4-bromo-aniline With hydrogenchloride in water 2: With sodium nitrite in water T=15°C; 3: chloroacetic acid ethyl ester With sodium acetate in ethanol; water T=20°C;
参考文献
Donohue, Sean R.; Dannals, Robert F.; Halldin, Christer; Pike, Victor W.
Journal of Medicinal Chemistry, 2011 , vol. 54, # 8 p. 2961 - 2970