反应条件
1: Et3N / CH2Cl2 / Ambient temperature 2: 1.) O3, 2.) H2O2 / 1.) Me2CO, water, 5 deg C, 30 min, 2.) Me2CO, water, 20 deg C, overnight View Scheme
参考文献
Ludeman; Boyd; Regan; Gallo; Zon; Ishii
Journal of Medicinal Chemistry, 1986 , vol. 29, # 5 p. 716 - 727