2-羟基吡啶-5-硼酸频哪醇酯合成路线 (共 2 条)
反应条件
tetrakis(triphenylphosphine) palladium(0); sodium carbonate in water; acetonitrile T=75°C; Suzuki coupling;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 21, # 19 p. 5774 - 5777
反应条件
potassium carbonate in acetonitrile T=50°C; 16 h; Sealed vial;
参考文献
WO2012/125893 A1, ;
Page/Page column 212-213 ;
WO 2012/125893 A1