1: carbon disulfide; benzylamine With sodium hydroxide in ethanol T=100°C; Microwave irradiation; 2: chloroacetic acid in ethanol T=100°C; 0.0833333 h; Microwave irradiation; 3: With hydrogenchloride in ethanol; water T=120°C; P=7500.75 Torr; 0.5 h; Microwave irradiation;
参考文献
Nitsche, Christoph; Schreier, Verena N.; Behnam, Mira A. M.; Kumar, Anil; Bartenschlager, Ralf; Klein, Christian D.
Journal of Medicinal Chemistry, 2013 , vol. 56, # 21 p. 8389 - 8403
Gil, Ana Martinez; Morera, Ana Castro; Perez, Maria Concepcion Martin; Cascon, Mercedes Alonso; Diaz, Isabel Dorronsoro; Munoz, Francisco Jose Moreno; Jurado, Francisco Wandosell
Patent: US2003/195238 A1, 2003 ;
Location in patent: Page/Page column 12 ;