反应条件
1: 1) NaH, 2) 2N aq. NaOH / 1) 150 deg C, 2 h, 2) MeOH, 20 deg C, 10 min 2: 1) N-hydroxysuccinimide, dicyclohexylcarbodiimide / 1) CHCl3, 3 h, 2) CHCl3, 25 deg C, 1 d 3: 2N NaOH / methanol View Scheme
参考文献
Journal of Medicinal Chemistry, , vol. 32, # 7 p. 1436 - 1441