1: 4-bromo-phenol With di-isopropyl azodicarboxylate; triphenylphosphine; Wang resin in tetrahydrofuran
T=20°C;
2: dihydroxy(3-fluorophenyl)borane With sodium carbonate; tetrakis(triphenylphosphine) palladium(0) in ethylene glycol dimethyl ether; water
T=80°C; Suzuki reaction;
3: With trifluoroacetic acid in dichloromethane
0.166667 h;
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