2-氯-5-碘-7H-吡咯并[2,3-d]嘧啶合成路线 (共 1 条)
反应条件
N-iodo-succinimide in acetonitrile T=12 - 20°C; 1 h;
参考文献
PFIZER LIMITED; ANDREWS, Mark, David; BAGAL, Sharanjeet, Kaur; BROWN, David, Graham; GIBSON, Karl, Richard; OMOTO, Kiyoyuki; RYCKMANS, Thomas; SABNIS, Yogesh; SKERRATT, Sarah, Elizabeth; STUPPLE, Paul, Anthony
Patent: WO2014/53967 A1, 2014 ;
Location in patent: Page/Page column 134 ;