(4S,5R)-5-[3,5-二(三氟甲基)苯基]-3-[[4'-氟-2'-(三氘甲氧基)-5'-(异丙基)-4-(三氟甲基)[1,1'-联苯]-2-基]甲基]-4-甲基-2-恶唑烷酮合成路线 (共 1 条)
反应条件
potassium carbonate in N,N-dimethyl-formamide T=20 - 60°C;
参考文献
CONCERT PHARMCEUTICALS, INC.
Patent: US2008/242711 A1, 2008 ;
Location in patent: Page/Page column 15-16 ;