反应条件
1: Et3N / CH2Cl2 / 0 °C 2: TMEDA, n-BuLi / diethyl ether; hexane / 1.) room temperature, 4 h, 2.) -5 deg C, 1 h View Scheme
参考文献
Adelstein, Gilbert W.; Yen, Chung H.; Haack, Richard A.; Yu, Stella; Gullikson, Gary; et al.
Journal of Medicinal Chemistry, 1988 , vol. 31, # 6 p. 1215 - 1220