反应条件
1: anthranilic acid With 1,1'-carbonyldiimidazole in N,N-dimethyl-formamide T=40°C; 2: propylamine in N,N-dimethyl-formamide T=20°C;
参考文献
Mizutani, Takashi; Nagase, Tsuyoshi; Ito, Sayaka; Miyamoto, Yasuhisa; Tanaka, Takeshi; Takenaga, Norihiro; Tokita, Shigeru; Sato, Nagaaki
Bioorganic and Medicinal Chemistry Letters, 2008 , vol. 18, # 23 p. 6041 - 6045