2-氨基-5-溴吡啶合成路线

参考文献

Ross Kelly; Jagoe; Gu
Tetrahedron Letters, 1991 , vol. 32, # 34 p. 4263 - 4266

1072-97-52-氨基-5-溴吡啶+

24424-99-5二碳酸二叔丁酯

209959-28-4+

159451-66-82-(Boc-氨基)-5-溴吡啶

参考文献

Bristol-Myers Squibb Pharma Company
Patent: EP946508 B1, 2009 ;
Location in patent: Page/Page column 59 ;

1072-97-52-氨基-5-溴吡啶+

171364-80-0对甲氧羰基苯硼酸频哪醇酯

222986-49-4

参考文献

Motiwala, Hashim; Kandre, Shivaji; Birar, Vishal; Kadam, Kishorkumar S.; Rodge, Atish; Jadhav, Ravindra D.; Mahesh Kumar Reddy; Brahma, Manoja K.; Deshmukh, Nitin J.; Dixit, Amol; Doshi, Lalit; Gupte, Amol; Gangopadhyay, Ashok K.; Vishwakarma, Ram A.; Srinivasan, Shaila; Sharma, Mamta; Nemmani, Kumar V.S.; Sharma, Rajiv
Bioorganic and Medicinal Chemistry Letters, 2011 , vol. 21, # 19 p. 5812 - 5817

1072-97-52-氨基-5-溴吡啶+

15568-86-25-乙氧基甲烯基-2,2-二甲基-1,3-二氧六环-4,6-二酮

25165-70-2

参考文献

Ravina; Zicane; Petrova; Gudriniece; Kalejs
Chemistry of Heterocyclic Compounds, 2002 , vol. 38, # 7 p. 836 - 839

1072-97-52-氨基-5-溴吡啶+

15568-85-15-(甲氧基甲烯基)-2,2-二甲基-1,3-二氧己环-4,6-二酮

25165-70-2

参考文献

Molnar, Annamaria; Faigl, Ferenc; Podanyi, Benjamin; Finta, Zoltan; Balazs, Laszlo; Hermecza, Istvan
Heterocycles, 2009 , vol. 78, # 10 p. 2477 - 2488

1072-97-52-氨基-5-溴吡啶

23536-76-77-溴-吡啶并[1,2-a]嘧啶-4-酮

参考文献

Ravina; Zicane; Petrova; Gudriniece; Kalejs
Chemistry of Heterocyclic Compounds, 2002 , vol. 38, # 7 p. 836 - 839

参考文献

Uckun, Fatih M.; Tibbles, Heather; Erbeck, Douglas; Venkatachalam, Taracad K.; Qazi, Sanjive
Arzneimittel-Forschung/Drug Research, 2007 , vol. 57, # 4 p. 218 - 226

1072-97-52-氨基-5-溴吡啶

870521-31-65-溴-2-异丙氧基吡啶

参考文献

Shibasaki
Yakugaku Zasshi, 1952 , vol. 72, p. 381
Chem.Abstr., 1953 , p. 6403

1072-97-52-氨基-5-溴吡啶+

1147550-11-5

31430-38-31-(5-溴-2-吡啶基)-2-硫脲

参考文献

MERCK PATENT GMBH
Patent: WO2009/46784 A1, 2009 ;
Location in patent: Page/Page column 49-50 ;
WO 2009/046784 A1

1072-97-52-氨基-5-溴吡啶+

1679-18-14-氯苯硼酸

84596-08-7

参考文献

F. HOFFMANN-LA ROCHE AG; BRUMSTED, Corey James; MOORLAG, Hendrik; RADINOV, Roumen Nikolaev; REN, Yi; WALDMEIER, Pius
Patent: WO2012/10538 A2, 2012 ;
Location in patent: Page/Page column 23 ;