2-(甲氧基羰基)-4-(三氟甲基)苯硼酸合成路线 (共 1 条)
反应条件
1: potassium carbonate / tetrakis(triphenylphosphine) palladium(0) / tetrahydrofuran / Reflux
2: lithium aluminium tetrahydride / diethyl ether / 10 h / Inert atmosphere; Reflux
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参考文献
ZHEJIANG BETA PHARMA INC.; KANG, Xinshan; LONG, Wei; WANG, Yanping; HU, Yunyan; WANG, Yinxiang
Patent: WO2012/41253 A1, 2012 ;
WO 2012/041253 A1