反应条件
4-(N,N-dimethlyamino)pyridine; triethylamine in pyridine; N,N-dimethyl-formamide T=80°C; 16 h; SolventTemperature;
参考文献
Merk, Daniel; Gabler, Matthias; Gomez, Roberto Carrasco; Flesch, Daniel; Hanke, Thomas; Kaiser, Astrid; Lamers, Christina; Werz, Oliver; Schneider, Gisbert; Schubert-Zsilavecz, Manfred
Bioorganic and Medicinal Chemistry, 2014 , vol. 22, # 8 p. 2447 - 2460