反应条件
1: 93 percent / 2,6-lutidine / CH2Cl2 / 24 h 2: 78 percent / aq. LiOH / tetrahydrofuran; methanol / 4 h 3: 7.4 percent / 1-<3-(dimethylamino)propyl>-3-ethylcarbodiimide hydrochloride, 4-(dimethylamino)pyridine / CH2Cl2 / 48 h View Scheme
参考文献
Matassa; Brown; Bernstein; Shapiro; Maduskuie Jr.; Cronk; Vacek; Yee; Snyder; Krell; Lerman; Maloney
Journal of Medicinal Chemistry, 1990 , vol. 33, # 9 p. 2621 - 2629
