反应条件
1: conc. HBr, HOAc / 1.25 h / 90 °C 2: 28 percent / toluene / Heating 3: 1.) NH3 (liq.), Na / 2.) MeOH, 45 deg C, 15 min View Scheme
参考文献
Graham, Donald W.; Ashton, Wallace T.; Barash, Louis; Brown, Jeannette E.; Brown, Ronald D.; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 6 p. 1074 - 1090
