反应条件
1: vinyl acetate; (1R,4S)-4-Azido-cyclopent-2-enol With Pancreatin in tetrahydrofuran Acetylation; 3 h; 2: di-tert-butyl dicarbonate With hydrogen; palladium on activated charcoal in ethyl acetate reductive acylation; P=3102.89 Torr; Title compound not separated from byproducts;
参考文献
Barrow, James C.; Glass, Kristen L.; Selnick, Harold G.; Freidinger, Roger M.; Chang, Raymond S.L.; O'Malley, Stacey S.; Woyden, Carla
Bioorganic and Medicinal Chemistry Letters, 2000 , vol. 10, # 17 p. 1917 - 1920