6-甲氧基-2-甲基-3-(4,4,5,5-四甲基-[1,3,2] 二噁硼烷-2-基)-吡啶合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in N,N-dimethyl-formamide T=80°C; 18 h; Product distribution / selectivity;
参考文献
VERTEX PHARMACEUTICALS INCORPORATED
Patent: WO2008/141119 A2, 2008 ;
Location in patent: Page/Page column 95-96; 99-100 ;
WO 2008/141119 A2