4-氯-6-甲基噻吩并[3,2-d]嘧啶合成路线 (共 1 条)
反应条件
1: 4-Chlorothieno[3,2-d]pyrimidine With sec.-butyllithium in tetrahydrofuran T=-78°C; 0.5 h; 2: methyl iodide in tetrahydrofuran T=20°C; 1 h;
参考文献
PFIZER INC.
Patent: WO2005/21553 A1, 2005 ;
Location in patent: Page/Page column 82-83 ;
WO 2005/021553 A1