反应条件
1: With triethylamine in N,N-dimethyl-formamide T=95 - 100°C; Leimgruber-Batcho Indole Synthesis; 4 h; Large scale; 2: With palladium 10 on activated carbon; hydrogen; sodium acetate in methanol; N,N-dimethyl-formamide T=30°C; Leimgruber-Batcho Indole Synthesis; 4 h; Large scale;
参考文献
Gillmore, Adam T.; Badland, Matthew; Crook, Clare L.; Castro, Nieves M.; Critcher, Douglas J.; Fussell, Steven J.; Jones, Katherine J.; Jones, Matthew C.; Kougoulos, Eleftherios; Mathew, Jinu S.; McMillan, Lynne; Pearce, John E.; Rawlinson, Fiona L.; Sherlock, Alexandra E.; Walton, Robert
Organic Process Research and Development, 2012 , vol. 16, # 12 p. 1897 - 1904
