3-碘-1H-吡唑并[3,4-c]吡啶合成路线 (共 1 条)
反应条件
iodine; potassium hydroxide in N,N-dimethyl-formamide T=20°C; 16 h;
参考文献
NOVARTIS AG; ALTMANN, Eva; HOMMEL, Ulrich; LORTHIOIS, Edwige Liliane Jeanne; MAIBAUM, Juergen Klaus; OSTERMANN, Nils; QUANCARD, Jean; RANDL, Stefan Andreas; VULPETTI, Anna
Patent: WO2014/2051 A2, 2014 ;
Location in patent: Page/Page column 54 ;