反应条件
1: pyridine / benzene / 70 °C 2: hydrogen, HOAc / 10percent Pd/C / hexane / 72 h / 2585.7 Torr 3: 45 percent / POCl3, Et3N / hexane; toluene / 18 h / Ambient temperature 4: 29 percent / pyridine / 120 h / Ambient temperature View Scheme
参考文献
Hong; An; Buchheit; Nechaev; Kirisits; West; Berdel
Journal of Medicinal Chemistry, 1986 , vol. 29, # 10 p. 2038 - 2044
