反应条件
1: 1.98 g / Ac2O / 2.5 h / 50 °C 2: 1.) NaH, DMSO / 1.) THF, 15 min, 2.) THF, 15 min View Scheme
参考文献
Milecki, Jan; Baker, Stephen P.; Standifer, Kelly M.; Ishizu, Takashi; Chida, Yasuhiro; et al.
Journal of Medicinal Chemistry, 1987 , vol. 30, # 9 p. 1563 - 1566