1: 7.0 g / NH4OAc; AcOH / 12 h / 20 °C
2: Pd(OAc)2; TEA; triethylsilane / CH2Cl2 / 3 h / 20 °C
View Scheme
参考文献
Bock, Mark G.; DiPardo, Robert M.; Evans, Ben E.; Rittle, Kenneth E.; Veber, Daniel F.; et al.
Journal of Organic Chemistry, 1987 , vol. 52, # 15 p. 3232 - 3239