GSK 1904529A; GSK 4529; N-(2,6-二氟苯基)-5-[3-[2-[[5-乙基-2-甲氧基-4-[4-[4-(甲基磺酰基)-1-哌嗪基]-1-哌啶基]苯基]氨基]-4-嘧啶基]咪唑并[1,2-a]吡啶-2-基]-2-甲氧基苯甲酰胺合成路线 (共 1 条)
反应条件
hydrogenchloride in 2,2,2-trifluoroethanol T=80 - 100°C; sealed vessel;
参考文献
Bioorganic and Medicinal Chemistry Letters, , vol. 19, # 3 p. 1004 - 1008