Chakrapani, Harinath; Kalathur, Ravi C.; Maciag, Anna E.; Citro, Michael L.; Ji, Xinhua; Keefer, Larry K.; Saavedra, Joseph E.
Bioorganic and Medicinal Chemistry, 2008 , vol. 16, # 22 p. 9764 - 9771
1: in butan-1-ol
T=0 - 20°C; 14 h;
2: With sodium hydroxide in water; toluene
pH=11.2;
3: With hydrogenchloride; sodium hydroxide
Product distribution / selectivity; more than 3 stages;
参考文献
Toray Fine Chemicals Co., Ltd.
Patent: EP1548010 A1, 2005 ;
Location in patent: Page/Page column 16; 20-21 ;