1: With hydrogenchloride in 1,4-dioxane T=20°C; 3 h; 2: With sodium hydrogencarbonate in water pH=8;
参考文献
MEDICAL RESEARCH COUNCIL TECHNOLOGY; MCIVER, Edward, Giles; HOUGH, Joane
Patent: WO2010/100431 A1, 2010 ;
Location in patent: Page/Page column 52 ;
WO 2010/100431 A1