6-甲氧基-[1,2,4]噻唑并[1,5-a]吡啶-2-胺合成路线 (共 2 条)
反应条件
hydroxylamine hydrochloride; N-ethyl-N,N-diisopropylamine in methanol; ethanol T=20 - 60°C; 6 h;
参考文献
US2009/270405 A1, ;
Page/Page column 81 ;
反应条件
1: 1,4-dioxane / 20 °C 2: hydroxylamine hydrochloride; N-ethyl-N,N-diisopropylamine / ethanol; methanol / 6 h / 20 - 60 °C View Scheme
参考文献
WO2011/53292 A1, ;
WO 2011/053292 A1