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乙二醇甲醛63148-62-9MDI丁酮二甲基亚砜碳酸氢钠471-34-1
AMG-221; (5S)-2-[(1S,2S,4R)-双环[2.2.1]庚烷-2-氨基]-5-甲基-5-异丙基-4(5H)-噻唑酮合成路线 (共 8 条)
参考文献
AMGEN INC.
Patent: WO2009/2445 A1, 2008 ;
Location in patent: Page/Page column 44-45 ;
WO 2009/002445 A1
参考文献
AMGEN INC.; CAILLE, Seb; CUI, Sheng; WANG, Silas; FAUL, Margaret
Patent: WO2010/14586 A1, 2010 ;
Location in patent: Page/Page column 24-25 ;
WO 2010/014586 A1
参考文献
Frizzle, Matthew J.; Nani, Roger R.; Martinelli, Michael J.; Moniz, George A.
Tetrahedron Letters, 2011 , vol. 52, # 43 p. 5613 - 5616
参考文献
AMGEN INC.; MONIZ, George A.; FRIZZLE, Matthew J.; BERNARD, Charles; MARTINELLI, Michael; FAUL, Margaret; LARROW, Jay; HANSEN, Karl B.; KLINGENSMITH, Liane
Patent: WO2010/8729 A2, 2010 ;
Location in patent: Page/Page column 45-46 ;
WO 2010/008729 A2
参考文献
AMGEN INC.; CAILLE, Seb; CUI, Sheng; WANG, Silas; FAUL, Margaret
Patent: WO2010/14586 A1, 2010 ;
Location in patent: Page/Page column 22 ;
WO 2010/014586 A1
参考文献
Frizzle, Matthew J.; Nani, Roger R.; Martinelli, Michael J.; Moniz, George A.
Tetrahedron Letters, 2011 , vol. 52, # 43 p. 5613 - 5616
参考文献
Veniant, Murielle M.; Hale, Clarence; Hungate, Randall W.; Gahm, Kyung; Emery, Maurice G.; Jona, Janan; Joseph, Smriti; Adams, Jeffrey; Hague, Andrew; Moniz, George; Zhang, Jiandong; Bartberger, Michael D.; Li, Vivian; Syed, Rashid; Jordan, Steven; Komorowski, Renee; Chen, Michelle M.; Cupples, Rod; Kim, Ki Won; St. Jean, David J.; Johansson, Lars; Henriksson, Martin A.; Williams, Meredith; Vallgarda, Jerk; Fotsch, Christopher; Wang, Minghan
Journal of Medicinal Chemistry, 2010 , vol. 53, # 11 p. 4481 - 4487
参考文献
AMGEN INC.
Patent: WO2009/2445 A1, 2008 ;
Location in patent: Page/Page column 46-47 ;
WO 2009/002445 A1