2-(叔丁氧基羰基氨基)吡啶-4-硼酸频那醇酯合成路线 (共 1 条)
反应条件
potassium acetate; (1,1'-bis(diphenylphosphino)ferrocene)palladium(II) dichloride in dimethyl sulfoxide T=85°C; 1.25 h; Inert atmosphere;
参考文献
PFIZER LIMITED; ICAGEN, INC.; GREENER, Benjamin Scott; MARRON, Brian Edward; MILLAN, David Simon; RAWSON, David James; STORER, Robert Ian; SWAIN, Nigel Alan
Patent: WO2012/4714 A2, 2012 ;
Location in patent: Page/Page column 62 ;
WO 2012/004714 A2