1: With diisobutylaluminium hydride in tetrahydrofuran
T=-78 - 40°C; 3 h;
2: With water; ammonium chloride in tetrahydrofuran
Product distribution / selectivity;
参考文献
Wyeth
Patent: US2009/18332 A1, 2009 ;
Location in patent: Page/Page column 14 ;
US 20090018332 A1