(4-羟基哌啶-1-基)-[4-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯基]甲酮合成路线 （共 1 条）
反应条件
1: 4-(4,4,5,5-tetramethyl-[1,3,2]dioxaborolan-2-yl)-benzoic acid With benzotriazol-1-ol; 1-ethyl-(3-(3-dimethylamino)propyl)-carbodiimide hydrochloride in N,N-dimethyl-formamide 4 h; 2: 4-hydroxy-piperidine in N,N-dimethyl-formamide
参考文献
ASTRAZENECA AB
Patent: WO2009/7390 A2, 2009 ;
Location in patent: Page/Page column 95 ;
WO 2009/007390 A2
