1: glycine With pyridine-2-carboxylic acid(2-benzoyl-phenyl)-amide; sodium methylate; nickel(II) nitrate hexahydrate in methanol 0.333333 h; Heating; 2: 3-fluoro-1-bromomethylbenzene With sodium hydroxide; (R)-NOBIN in dichloromethane T=20°C; 0.116667 h; 3: With hydrogenchloride in methanol; water Heating;
参考文献
Angewandte Chemie - International Edition, , vol. 40, # 10 p. 1948 - 1951