反应条件
1: 1.) Mg / 1.) THF, 30 deg C, 2 h, 2.) THF, from -80 deg C to RT, overnight 2: 11 percent / 48percent aq. HBr / Heating View Scheme
参考文献
Mirabelli; Hill; Faucette; McCabe; Girard; Bryan; Sutton; O'Leary Bartus; Crooke; Johnson
Journal of Medicinal Chemistry, 1987 , vol. 30, # 12 p. 2181 - 2190