6-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)苯并[d]异噻唑合成路线 (共 1 条)
反应条件
potassium acetate; tri-cyclo-hexyl-phosphine; tris-(dibenzylideneacetone)dipalladium(0) in 1,4-dioxane T=110°C; 0.5 h; Sealed tubeMicrowave irradiation;
参考文献
AMGEN INC.
Patent: WO2009/11871 A2, 2009 ;
Location in patent: Page/Page column 185 ;
WO 2009/011871 A2