1-甲基-5-(4,4,5,5-四甲基-1,3,2-二硼戊环-2-基)-1H-苯并[d]咪唑合成路线 (共 1 条)
反应条件
dichloro(1,1'-bis(diphenylphosphanyl)ferrocene)palladium(II) dichloromethane adduct; potassium acetate in 1,4-dioxane T=160°C; 0.333333 h; Inert atmosphereMicrowave irradiation;
参考文献
TAKEDA PHARMACEUTICAL COMPANY LIMITED; LAWSON, John David; SABAT, Mark; SMITH, Christopher; WANG, Haixia; CHEN, Young K.; KANOUNI, Toufike
Patent: WO2013/148603 A1, 2013 ;
Location in patent: Paragraph 0219-0220 ;