反应条件
1: 95 percent / piperidine, AcOH / toluene / 3.5 h / Heating 2: H2, Et3N / 10percent Pd/C / Ambient temperature 3: 1.) CF3COOH / 1.) 10 min, 2.) 0 deg C, 10 min View Scheme
参考文献
Smith, Kevin M.; Pandey, Ravindra K.; Tabba, Hani D.
Journal of Chemical Research, Miniprint, 1986 , # 11 p. 3333 - 3357