Kirpichenok, M. A.; Mel'nikova, L. M.; Denisov, L. K.; Grandberg, I. I.
Chemistry of Heterocyclic Compounds (New York, NY, United States), 1988 , vol. 24, # 9 p. 959 - 965
Khimiya Geterotsiklicheskikh Soedinenii, 1988 , # 9 p. 1169 - 1175
1: With 1,3-bis-(diphenylphosphino)propane; potassium carbonate; palladium diacetate in DMF (N,N-dimethyl-formamide); water T=20 - 80°C; 24 h; 2: With formic acid; water in acetonitrile T=20°C; 0.75 h;
参考文献
GLAXO GROUP LIMITED
Patent: WO2004/110997 A1, 2004 ;
Location in patent: Page 52-53 ;
WO 2004/110997 A1
1: With 1,3-bis-(diphenylphosphino)propane; triethylamine; palladium diacetate in various solvent(s) T=125°C; Regioselective Heck arylation; 30 h; 2: With hydrogenchloride in various solvent(s) 1 h;
参考文献
Pei, Wen; Mo, Jun; Xiao, Jianliang
Journal of Organometallic Chemistry, 2005 , vol. 690, # 15 p. 3546 - 3551
