N,3-二甲基-5-(4,4,5,5-四甲基-1,3,2-二噁硼烷-2-基)吡啶-2-胺合成路线 (共 1 条)
反应条件
potassium acetate; bis-triphenylphosphine-palladium(II) chloride in N,N-dimethyl-formamide
T=80 - 90°C;
参考文献
PFIZER INC.
Patent: WO2009/16460 A2, 2009 ;
Location in patent: Page/Page column 65-66 ;
WO 2009/016460 A2