反应条件
1: 97 percent / POCl3, N,N-dimethylaniline / Heating 2: 82 percent / NH3(g) / dimethylformamide / 0.67 h / 35 - 40 °C 3: 59.7 percent / butan-1-ol / 14 h / 95 °C View Scheme
参考文献
Volzhina, O. N.; Azimov, V. A.; Medvedev, B. A.; Kazakov, A. A.; Zhikhareva, G. P.; et al.
Pharmaceutical Chemistry Journal, 1987 , vol. 21, # 7 p. 478 - 483
Khimiko-Farmatsevticheskii Zhurnal, 1987 , vol. 21, # 7 p. 802 - 807