1-(2-嘧啶基)哌啶-4-甲酸乙酯合成路线 (共 2 条)
反应条件
triethylamine in toluene Heating;
参考文献
Cignarella; Villa; Barlocco
Farmaco, 1993 , vol. 48, # 10 p. 1439 - 1445
反应条件
lithium hydroxide hydrate; water in tetrahydrofuran T=20°C; 18 h; Inert atmosphere;
参考文献
VANTIA LIMITED; BATT, Andrzej, Roman; HEENEY, Celine, Marguerite, Simone
Patent: WO2010/97576 A1, 2010 ;
Location in patent: Page/Page column 43-44 ;
WO 2010/097576 A1