6-溴-8-三氟甲基吲唑并[1,2-A]吡啶-2-甲酸乙酯合成路线 (共 1 条)
反应条件
in N,N-dimethyl-formamide T=50°C; 24 h;
参考文献
GLAXOSMITHKLINE LLC; BANKA, Anna; BASKARAN, Subramanian; CATALANO, John; CHONG, Pek; DICKSON, Hamilton; FANG, Jing; MAUNG, Jack; NEITZEL, Martin, Leon; PEAT, Andy; PRICE, Daniel; RAI, Roopa; ROBERTS, Christopher, Don; SHOTWELL, Brad; TAI, Vincent; ZHANG, Huichang
Patent: WO2010/91411 A1, 2010 ;
Location in patent: Page/Page column 79 ;
WO 2010/091411 A1